Signaling signature of neurotensin receptor type 1 with endogenous ligands. Besserer-Offroy É, Brouillette RL, Lavenus S, Froehlich U, Brumwell A, Murza A, Longpré JM, Marsault É, Grandbois M, Sarret P, Leduc R. Eur J Pharmacol. 2017 Mar 21. doi: 10.1016/j.ejphar.2017.03.046
New manuscript accepted in Organic and Biomolecular Chemistry
Structure-activity relationship of novel macrocyclic biased apelin receptor agonists. Murza A, Sainsily X, Côté J, Bruneau-Cossette L, Besserer-Offroy É, Longpré JM, Leduc R, Dumaine R, Lesur O, Auger-Messier M, Sarret P, Marsault É. Org Biomol Chem. 2016 Dec 7. PMID: 27924341
Presentation prize at Journée Phare 2016
I have been selected for a talk at Journée Phare 2016 and my presentation “Phosphomimetic lipopeptides as new tools to investigate β-arrestin-mediated functions.” won the second best oral presentation !
Manuscript accepted in Organic and Biomolecular Chemistry
Design, Synthesis, and Biological Evaluation of Novel CXCR4 Inverse Agonists Mona CE, Besserer-Offroy É, Cabana J, Leduc R, Lavigne P, Heveker N, Marsault E, Escher E Org Biomol Chem. 2016 Oct 04. DOI: 10.1039/C6OB01484D
Abstract for Neuroscience 2016 is now online
My abstract, “Phosphomimetic lipopeptides as new tools to investigate β-arrestin-mediated functions.” which has been selected for presentation in a nanosymposium at Neuroscience 2016 is now online. Click here to view it. Here are the details for the nanosymposium: Molecular Techniques (session # 673) Wednesday Nov 16, 2016 – from 8:00 AM to 12:00 PM San […]
Manuscript accepted in the Journal of Medicinal Chemistry
Structure Activity Relationship and Signaling of New Chimeric CXCR4 Agonists. Mona CE, Besserer-Offroy É, Cabana J, Lefrançois M, Boulais PE, Lefebvre MR, Leduc R, Lavigne P, Heveker N, Marsault E, Escher E. J Med Chem. 2016 Jul 19. PMID: 27434274
Abstract accepted for Nanosymposium presentation at Neuroscience 2016 in San Diego
My abstract, “Phosphomimetic lipopeptides as new tools to investigate β-arrestin-mediated functions.” has been selected for presentation in a nanosymposium at the 2016 Annual Meeting of the Society for Neuroscience in San Diego, California. Here are the details for the nanosymposium: Molecular Techniques (session # 673) Wednesday Nov 16, 2016 – from 8:00 AM to 12:00 […]
Manuscript accepted in ACS Chemical Neuroscience
Identification of 2-({[1-(4-fluorophenyl)-5-(2-methoxyphenyl)-1H-pyrazol-3-yl]carbonyl}amino)tricyclo[3.3.1.13,7]decane-2-carboxylic acid (NTRC-844) as a selec-tive antagonist for the Rat Neurotensin recep-tor type 2. Thomas JB, Vivancos M, Giddings AM, Wiethe RW, Warner KR, Murza A, Besserer-Offroy É, Longpre JM, Runyon SP, Decker AM, Gilmour BP, Sarret P. ACS Chem Neurosci. 2016 Jun 30. PMID: 27359371
Canadian Student Health Research Forum 2016
I have been nominated to represent the Université de Sherbrooke at the 2016 edition of the Canadian Student Health Research Forum held at Winnipeg (MB) on June 7-9, 2016 (as being in the top 5% of doctoral students in Canada). I also received a Travel grant from the Canadian Institutes of Health Research ($1,000) to attend […]
Manuscript accepted in the Journal of Medicinal Chemistry
Discovery and structure-activity relationship of a bioactive fragment of ELABELA that modulates vascular and cardiac functions. Murza A, Sainsily X, Coquerel D, Côté J, Marx P, Besserer-Offroy É, Longpre JM, Lainé J, Reversade B, Salvail D, Leduc R, Dumaine R, Lesur O, Auger-Messier M, Sarret P, Marsault E. J Med Chem. 2016 Mar 17. PMID: […]